UPF 1069

CAS No. 1048371-03-4

UPF 1069 ( UPF-1069, UPF1069, UPF 1069 )

Catalog No. M17125 CAS No. 1048371-03-4

UPF 1069 is a specific PARP2 inhibitor ( IC50: 0.3 μM). It is ~27-fold selective against PARP1.

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 38 In Stock
10MG 59 In Stock
25MG 113 In Stock
50MG 177 In Stock
100MG 296 In Stock
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Biological Information

  • Product Name
    UPF 1069
  • Note
    Research use only, not for human use.
  • Brief Description
    UPF 1069 is a specific PARP2 inhibitor ( IC50: 0.3 μM). It is ~27-fold selective against PARP1.
  • Description
    UPF-1069 is a selective and potent PARP2 inhibitor. UPF-1069 induces apoptosis. UPF-1069 shows neuroprotective and anti-ischemic effects in vivo.
  • Synonyms
    UPF-1069, UPF1069, UPF 1069
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    PARP1; PARP2
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    1048371-03-4
  • Formula Weight
    279.29
  • Molecular Formula
    C17H13NO3
  • Purity
    98%
  • Solubility
    DMSO : ≥ 100 mg/mL 358.05 mM
  • SMILES
    c1(=O)[nH]ccc2c(cccc12)OCC(=O)c1ccccc1
  • Chemical Name
    5-(2-oxo-2-phenylethoxy)isoquinolin-1(2H)-one

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Moroni F, et al. Br J Pharmacol, 2009, 157(5), 854-862.
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